首页>新闻资讯 2025-06-06 16:23:07
Bupivacaine-d9,布比卡因-d9「同位素标记抑制剂」
生物活性:Bupivacaine-d99 is a deuterium labeled Bupivacaine. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain[1][2][3].
IC50 & Target:NMDA Receptor
分子量:297.48
Formula:C18H19D9N2O
CAS 号:474668-57-0
非标记 CAS:38396-39-3
性状:固体
颜色:White to off-white
中文名称:布比卡因-d9
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month
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