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「同位素标记抑制剂」CAS:2714485-49-9|Verapamil-d3 hydrochloride
生物活性:Verapamil-d3 (hydrochloride) is the deuterium labeled Verapamil hydrochloride. Verapamil hydrochloride ((±)-Verapamil hydrochloride) is a calcium channel blocker and a potent and orally active first-generation P-glycoprotein (P-gp) inhibitor. Verapamil hydrochloride also inhibits CYP3A4. Verapamil hydrochloride has the potential for high blood pressure, heart arrhythmias and angina research[1][2][3].
体外研究(In Vitro):Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
德尔塔生物 has not independently confirmed the accuracy of these methods. They are for reference only.
Verapamil-d3 hydrochloride 相关抗体:
Annexin VI Antibody
Cytochrome C Antibody
Calbindin Antibody
Calreticulin Antibody
Cytochrome P450 17A1 Antibody
Aromatase Antibody
P Glycoprotein Antibody
Cardiac Troponin I/TNNC1 Antibody
CYP11A1 Antibody
SCGN Antibody (YA1167)
MRP1 Antibody (YA1583)
RAMP1 Antibody (YA1818)
Annexin V Antibody (YA1829)
Cytochrome P450 1B1 Antibody (YA1836)
Adrenodoxin Antibody (YA2005)
Striatin 4 Antibody (YA2088)
Cytochrome P450 27A1 Antibody (YA2163)
Cytochrome P450 2C9 Antibody (YA2166)
Cytochrome P450 2E1 Antibody (YA2302)
Fibulin 5 Antibody (YA2448)
RASGRP1 Antibody (YA2546)
Cytochrome P450 Reductase Antibody (YA2619)
Thromboxane A Synthase Antibody (YA2670)
Fibulin 1 Antibody (YA2831)
EFEMP1 Antibody (YA2883)
CRCP Antibody (YA3350)
Cytochrome P450 3A4 Antibody (YA3365)
HSD11B1 Antibody (YA3376)
Cytochrome P450 17A1 Antibody (YA786)
CYP2E1 Antibody
分子量:494.08
Formula:C27H36D3ClN2O4
CAS 号:2714485-49-9
非标记 CAS:152-11-4
性状:固体
颜色:White to off-white
中文名称:盐酸维拉帕米 d3 (盐酸盐)
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:4°C, sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
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