生物活性：Apremilast-d5 is a deuterium labeled Apremilast. Apremilast is an orally available inhibitor of type-4 cyclic nucleotide phosphodiesterase (PDE-4) with an IC50 of 74 nM. Apremilast inhibits TNF-α release by lipopolysaccharide (LPS) with an IC50 of 104 nM[1].
IC50 & Target[1]：PDE4
分子量：465.53
Formula：C22H19D5N2O7S
CAS 号：1258597-47-5
非标记 CAS：608141-41-9
性状：固体
颜色：Off-white to light yellow
中文名称：阿普司特 d5
运输条件：Room temperature in continental US; may vary elsewhere.
储存方式：Powder：-20°C：3 years，4°C：2 years
In solvent：-80°C：6 months，-20°C：1 month