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「同位素标记抑制剂」CAS:1127253-02-4|Prasugrel-d3
生物活性:Prasugrel-d3 is the deuterium labeled Prasugrel. Prasugrel (PCR 4099), a thienopyridine and proagent, inhibits platelet function. Prasugrel is an orally active and potent P2Y12 receptor antagonist, and inhibits ADP-induced platelet aggregation[1].
IC50 & Target:P2Y12 Receptor
体外研究(In Vitro):氢、碳和其他元素的稳定重同位素已被掺入药物分子中,主要用作药物开发过程中定量的示踪剂。氘代因其可能影响药物的药代动力学和代谢特征而受到关注[1]。
德尔塔生物 has not independently confirmed the accuracy of these methods. They are for reference only.
Prasugrel-d3 相关抗体:
P2Y12 Antibody (YA3135)
P2Y6 Antibody (YA1691)
分子量:376.46
Formula:C20H17D3FNO3S
CAS 号:1127253-02-4
非标记 CAS:150322-43-3
性状:固体
颜色:White to off-white
中文名称:普拉格雷 d3
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years,4°C:2 years
In solvent:-80°C:6 months,-20°C:1 month
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