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「同位素标记抑制剂」CAS:1216745-79-7|Mefenamic acid-d4
生物活性:Mefenamic acid-d4 is a deuterium labeled Mefenamic acid. Mefenamic acid is a non-steroidal anti-inflammatory agent, acting as a competitive inhibitor of hCOX-1 and hCOX-2, with IC50s of 40 nM and 3 μM for hCOX-1 and hCOX-2, respectively[1][2].
IC50 & Target:hCOX-1
40 nM (IC50)
hCOX-2
3 nM (IC50)
分子量:245.31
Formula:C15H11D4NO2
CAS 号:1216745-79-7
非标记 CAS:61-68-7
性状:固体
颜色:White to off-white
中文名称:甲芬那酸 d4
运输条件:Room temperature in continental US; may vary elsewhere.
储存方式:Powder:-20°C:3 years
In solvent:-80°C:6 months,-20°C:1 month
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